Product Details
Molecular Formula: C36H39N3O6 ∙ HCl
Formula Weight: 609.72 ∙ 36.46
CAS Number: 119934-51-9
Purity: >98%
Formulation: powder
Solubility: Soluble in DMSO (up to 25 mg/ml) or in Methanol (up to 25 mg/ml).
Storage: RT
Stability: ≥ 1 year.
Applications
L-type Ca2+ channel blocker
Functions
L-type calcium channel blocker (IC50 = 75 nM), which can also inhibit T-type calcium channels at higher concentrations (IC50 = 244 nM). Novel inhibitor of drug transport by p-glycoprotein.
Application Procedures
First dissolved in DMSO (up to 25 mg/ml) or in Methanol (up to 25 mg/ml), then diluted to aqueous buffer. Solutions in DMSO or methanol may be stored at -20°C for up to 3 months.