Tribioscience BML-259, CDK5/p25 Inhibitor (TBI1025)
SKU: TBI1025-5MG
Tribioscience BML-259, CDK5/p25 Inhibitor (TBI1025)
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Product Details
Formal Name: N-(5-isopropyl-thiazol-2-yl)phenylacetamide
Molecular Formula: C14H16N2OS
Formula Weight: 260.36
CAS Number: 267654-00-2
Purity: >98%
Formulation: powder
Solubility: Soluble in DMSO (up to 25 mg/ml).
Storage: RT
Stability: ≥ 1 year.
Applications
CDK5/p25 inhibitor
Functions
Potent inhibitor of Cdk5/p25 (IC50 = 64 nM) and Cdk2 (IC50 = 98nM).
Application Procedures
First dissolved in DMSO (up to 25 mg/ml), then diluted to aqueous buffer. Solutions in DMSO may be stored at -20°C for up to 3 months.